333 |
Lukin, A.; Komarova, K.; Vinogradova, L.; Rogacheva, E.; Kraeva, L.; Krasavin, M. Synthesis and antibacterial evaluation of ciprofloxacin congeners with spirocyclic amine periphery. Int. J. Mol. Sci. 2023, 24, 954 |
332 |
Dar'in, D.; Kantin, G.; Glushakova, D.; Sharoyko, V.; Krasavin, M. Diazo Tetramic Acids Provide Access to Natural-Like Spirocyclic Δα,β-Butenolides through Rh(II)-catalyzed O-H Insertion/Base-Promoted Cyclization. J. Org. Chem., accepted 26.12.2022 |
331 |
Krivovicheva, V.; Bubyrev, A.; Kalinin, S.; Dar'in, D.; Gureev, M.; Vullo, D.; Krasavin, M.; Korsakov, M.; Supuran, C. T. A new way of synthesizing heterocyclic primary sulfonamide probes for carbonic anhydrase. Mendeleev Commun., accepted 23.12.2022 |
330 |
Krasavin, M.; Adamchik, M.; Bubyrev, A.; Heim, C.; Maiwald, S.; Zhukovsky, D.; Zhmurov, P.; Bunev, A.; Hartmann, M. D. Synthesis of novel glutarimide ligands for the E3 ligase substrate receptor Cereblon (CRBN): investigation of their binding mode and antiproliferative effects against myeloma cell lines. Eur. J. Med. Chem. 2023, 246, 114990 |
329 |
Lukin, A.; Vinogradova, L.; Komarova, K.; Krasavin, M. Spirocyclic azetidines for drug discovery: novel Boc-protected 7'H-spiro[azetidine-3,5'-furo[3,4-d]pyrimidines]. Mendeleev Commun. 2022, accepted 10.11.2022 |
328 |
Lukin, A.; Vinogradova, L.; Komarova, K.; Kalinin, S.; Krasavin, M. Synthesis of 1-oxa-9-azaspiro[5.5]undecane-9-sulfonamides bearing a diverse molecular periphery and a rare zinc-binding group for carbonic anhydrase interrogation. Mendeleev Commun., accepted 01.11.2022 |
327 |
Solovyev, I.; Dar'in, D.; Krasavin, M. Synthetic enabling of spirocyclic oxetane fatty acid mimetics based on 1-oxa-6,7-diazaspiro[3.4]oct-7-en-5-one scaffold via diazo chemistry. Mendeleev Commun. 2023, 33, 21-23 |
326 |
Lukin, A.; Komarova, K.; Vinogradova, L.; Rogacheva, E.; Kraeva, L.; Dogonadze, M.; Vinogradova, T.; Krasavin, M. Urea derivatives of spirocyclic piperidines endowed with antibacterial activity. Mendeleev Commun. 2023, 33, 109-111 |
325 |
Adamchik, M.; Bubyrev, A.; Zhukovsky, D.; Zhmurov, P.; Bunev, A.; Krasavin, M. Synthesis of novel glutarimide derivatives via the Michael addition of (hetero)aromatic thiols: pronounced effect of sulfur oxidation on cytotoxicity towards multiple myeloma cell lines. Mendeleev Commun. 2023, 33, 67-69 |
324 |
Sibinčić, N.; Kalinin, S.; Sharoyko, V.; Efimova, J.; Gasilina, O. A.; Korsakov, M.; Gureev, M.; Krasavin, M. A Series of Trifluoromethylisoxazolyl- and Trifluoromethylpyrazolyl-Substituted (Hetero)aromatic Sulfonamide Carbonic Anhydrase Inhibitors: Synthesis and Convenient Prioritization Workflow for Further In Vivo studies. Med. Chem. 2023, 19, 193-210 |